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Discovery, oral pharmacokinetics and in vivo efficacy of velusetrag, a highly selective 5-HT(4) receptor agonist that has achieved proof-of-concept in patients with chronic idiopathic constipation. [electronic resource] by
- Long, Daniel D
- Armstrong, Scott R
- Beattie, David T
- Choi, Seok-Ki
- Fatheree, Paul R
- Gendron, Roland A L
- Genov, Daniel
- Goldblum, Adam A
- Humphrey, Patrick P
- Jiang, Lan
- Marquess, Daniel G
- Shaw, Jeng-Pyng
- Smith, Jacqueline A M
- Turner, S Derek
- Vickery, Ross G
Producer: 20130204
In:
Bioorganic & medicinal chemistry letters vol. 22
Availability: No items available.
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Synthesis and structure-activity relationship studies in serotonin 5-HT4 receptor ligands based on a benzo[de][2,6]naphthridine scaffold. [electronic resource] by
- Castriconi, Federica
- Paolino, Marco
- Giuliani, Germano
- Anzini, Maurizio
- Campiani, Giuseppe
- Mennuni, Laura
- Sabatini, Chiara
- Lanza, Marco
- Caselli, Gianfranco
- De Rienzo, Francesca
- Menziani, Maria Cristina
- Sbraccia, Maria
- Molinari, Paola
- Costa, Tommaso
- Cappelli, Andrea
Producer: 20150330
In:
European journal of medicinal chemistry vol. 82
Availability: No items available.
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