Results
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101.
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Discovery of Potent and Selective Inhibitors of Cdc2-Like Kinase 1 (CLK1) as a New Class of Autophagy Inducers. [electronic resource] by
- Sun, Qi-Zheng
- Lin, Gui-Feng
- Li, Lin-Li
- Jin, Xi-Ting
- Huang, Lu-Yi
- Zhang, Guo
- Yang, Wei
- Chen, Kai
- Xiang, Rong
- Chen, Chong
- Wei, Yu-Quan
- Lu, Guang-Wen
- Yang, Sheng-Yong
Producer: 20170905
In:
Journal of medicinal chemistry vol. 60
Availability: No items available.
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102.
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A preclinical evaluation of a novel multikinase inhibitor, SKLB-329, as a therapeutic agent against hepatocellular carcinoma. [electronic resource] by
- Zhong, Lei
- Fu, Xiao-Yu
- Zou, Chan
- Yang, Ling-Ling
- Zhou, Shu
- Yang, Jiao
- Tang, Yun
- Cheng, Chuan
- Li, Lin-Li
- Xiang, Rong
- Chen, Li-Juan
- Chen, Yu-Zong
- Wei, Yu-Quan
- Yang, Sheng-Yong
Producer: 20141209
In:
International journal of cancer vol. 135
Availability: No items available.
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103.
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Preclinical Evaluation of a Novel Orally Available SRC/Raf/VEGFR2 Inhibitor, SKLB646, in the Treatment of Triple-Negative Breast Cancer. [electronic resource] by
- Zheng, Ming-Wu
- Zhang, Chun-Hui
- Chen, Kai
- Huang, Mei
- Li, Ya-Ping
- Lin, Wan-Ting
- Zhang, Rong-Jie
- Zhong, Lei
- Xiang, Rong
- Li, Lin-Li
- Liu, Xin-Yu
- Wei, Yu-Quan
- Yang, Sheng-Yong
Producer: 20161213
In:
Molecular cancer therapeutics vol. 15
Availability: No items available.
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104.
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Structural optimization and structure-activity relationships of N2-(4-(4-Methylpiperazin-1-yl)phenyl)-N8-phenyl-9H-purine-2,8-diamine derivatives, a new class of reversible kinase inhibitors targeting both EGFR-activating and resistance mutations. [electronic resource] by
- Yang, Jiao
- Wang, Li-Jiao
- Liu, Jing-Jing
- Zhong, Lei
- Zheng, Ren-Lin
- Xu, Yong
- Ji, Pan
- Zhang, Chun-Hui
- Wang, Wen-Jing
- Lin, Xing-Dong
- Li, Lin-Li
- Wei, Yu-Quan
- Yang, Sheng-Yong
Producer: 20130226
In:
Journal of medicinal chemistry vol. 55
Availability: No items available.
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105.
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A novel orally available Syk/Src/Jak2 inhibitor, SKLB-850, showed potent anti-tumor activities in B cell lymphoma (BCL) models. [electronic resource] by
- Zhang, Nannan
- Zhang, Guo
- Liu, Ning
- Lin, Wanting
- Ji, Sen
- Zheng, Mingwu
- Chen, Kai
- Liang, Xiao
- Li, Guobo
- Ma, Yu
- Zhu, Jun
- Niu, Ting
- Li, Lin-Li
- Li, Jiong
- Wei, Yu-Quan
- Yang, Sheng-Yong
Publication details: Oncotarget Dec 2017
In:
Oncotarget vol. 8
Availability: No items available.
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106.
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Novel ROR1 inhibitor ARI-1 suppresses the development of non-small cell lung cancer. [electronic resource] by
- Liu, Xuesha
- Pu, Wenchen
- He, Huaiyu
- Fan, Xin
- Zheng, Yuanyuan
- Zhou, Jian-Kang
- Ma, Rui
- He, Juan
- Zheng, Yuzhu
- Wu, Ke
- Zhao, Yun
- Yang, Sheng-Yong
- Wang, Chun
- Wei, Yu-Quan
- Wei, Xia-Wei
- Peng, Yong
Producer: 20200528
In:
Cancer letters vol. 458
Availability: No items available.
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107.
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Accumulation of FLT3(+) CD11c (+) dendritic cells in psoriatic lesions and the anti-psoriatic effect of a selective FLT3 inhibitor. [electronic resource] by
- Yan, Heng-Xiu
- Li, Wei-Wei
- Zhang, Yan
- Wei, Xia-Wei
- Fu, Li-Xin
- Shen, Guo-Bo
- Yin, Tao
- Li, Xiu-Ying
- Shi, Hua-Shan
- Wan, Yang
- Zhang, Qing-Yin
- Li, Jiong
- Yang, Sheng-Yong
- Wei, Yu-Quan
Producer: 20150609
In:
Immunologic research vol. 60
Availability: No items available.
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108.
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Taking quinazoline as a general support-Nog to design potent and selective kinase inhibitors: application to FMS-like tyrosine kinase 3. [electronic resource] by
- Li, Wei-Wei
- Chen, Jin-Juan
- Zheng, Ren-Lin
- Zhang, Wen-Qin
- Cao, Zhi-Xing
- Yang, Ling-Ling
- Qing, Xiao-Yu
- Zhou, Liang-Xue
- Yang, Li
- Yu, Luo-Ding
- Chen, Li-Juan
- Wei, Yu-Quan
- Yang, Sheng-Yong
Producer: 20100708
In:
ChemMedChem vol. 5
Availability: No items available.
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109.
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Novel thienopyridine derivatives as specific anti-hepatocellular carcinoma (HCC) agents: synthesis, preliminary structure-activity relationships, and in vitro biological evaluation. [electronic resource] by
- Zeng, Xiu-Xiu
- Zheng, Ren-Lin
- Zhou, Tian
- He, Hai-Yun
- Liu, Ji-Yan
- Zheng, Yu
- Tong, Ai-Ping
- Xiang, Ming-Li
- Song, Xiang-Rong
- Yang, Sheng-Yong
- Yu, Luo-Ting
- Wei, Yu-Quan
- Zhao, Ying-Lan
- Yang, Li
Producer: 20110124
In:
Bioorganic & medicinal chemistry letters vol. 20
Availability: No items available.
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110.
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Drug Discovery against Psoriasis: Identification of a New Potent FMS-like Tyrosine Kinase 3 (FLT3) Inhibitor, 1-(4-((1H-Pyrazolo[3,4-d]pyrimidin-4-yl)oxy)-3-fluorophenyl)-3-(5-(tert-butyl)isoxazol-3-yl)urea, That Showed Potent Activity in a Psoriatic Animal Model. [electronic resource] by
- Li, Guo-Bo
- Ma, Shuang
- Yang, Ling-Ling
- Ji, Sen
- Fang, Zhen
- Zhang, Guo
- Wang, Li-Jiao
- Zhong, Jie-Min
- Xiong, Yu
- Wang, Jiang-Hong
- Huang, Shen-Zhen
- Li, Lin-Li
- Xiang, Rong
- Niu, Dawen
- Chen, Ying-Chun
- Yang, Sheng-Yong
Producer: 20170612
In:
Journal of medicinal chemistry vol. 59
Availability: No items available.
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111.
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SKLB610: a novel potential inhibitor of vascular endothelial growth factor receptor tyrosine kinases inhibits angiogenesis and tumor growth in vivo. [electronic resource] by
- Cao, Zhi-Xing
- Zheng, Ren-Lin
- Lin, Hong-Jun
- Luo, Shi-Dong
- Zhou, Yan
- Xu, You-Zhi
- Zeng, Xiu-Xiu
- Wang, Zhao
- Zhou, Li-Na
- Mao, Yong-Qiu
- Yang, Li
- Wei, Yu-Quan
- Yu, Luo-Ting
- Yang, Sheng-Yong
- Zhao, Ying-Lan
Producer: 20111003
In:
Cellular physiology and biochemistry : international journal of experimental cellular physiology, biochemistry, and pharmacology vol. 27
Availability: No items available.
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112.
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SKLB1206, a novel orally available multikinase inhibitor targeting EGFR activating and T790M mutants, ErbB2, ErbB4, and VEGFR2, displays potent antitumor activity both in vitro and in vivo. [electronic resource] by
- Pan, Youli
- Xu, Yong
- Feng, Shan
- Luo, Shidong
- Zheng, Renlin
- Yang, Jiao
- Wang, Lijiao
- Zhong, Lei
- Yang, Han-Yu
- Wang, Bing-Lin
- Yu, Yang
- Liu, Jingjing
- Cao, Zhixing
- Wang, Xiaoyan
- Ji, Pan
- Wang, Zerong
- Chen, Xin
- Zhang, Shuang
- Wei, Yu-Quan
- Yang, Sheng-Yong
Producer: 20121016
In:
Molecular cancer therapeutics vol. 11
Availability: No items available.
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113.
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Inhibition of Stat3 signaling pathway by nifuroxazide improves antitumor immunity and impairs colorectal carcinoma metastasis. [electronic resource] by
- Ye, Ting-Hong
- Yang, Fang-Fang
- Zhu, Yong-Xia
- Li, Ya-Li
- Lei, Qian
- Song, Xue-Jiao
- Xia, Yong
- Xiong, Ying
- Zhang, Li-Dan
- Wang, Ning-Yu
- Zhao, Li-Feng
- Gou, Hong-Feng
- Xie, Yong-Mei
- Yang, Sheng-Yong
- Yu, Luo-Ting
- Yang, Li
- Wei, Yu-Quan
Producer: 20171026
In:
Cell death & disease vol. 8
Availability: No items available.
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114.
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Structural optimization and structure-activity relationship studies of N-phenyl-7,8-dihydro-6H-pyrimido[5,4-b][1,4]oxazin-4-amine derivatives as a new class of inhibitors of RET and its drug resistance mutants. [electronic resource] by
- Yang, Jiao
- Chen, Kai
- Zhang, Guo
- Yang, Qiu-Yuan
- Li, Yue-Shan
- Huang, Shen-Zhen
- Wang, Yan-Lin
- Yang, Wei
- Jiang, Xiao-Juan
- Yan, Heng-Xiu
- Zhu, Jing-Qiang
- Xiang, Rong
- Luo, You-Fu
- Li, Wei-Min
- Wei, Yu-Quan
- Li, Lin-Li
- Yang, Sheng-Yong
Producer: 20180101
In:
European journal of medicinal chemistry vol. 143
Availability: No items available.
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115.
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Correction: Inhibition of Stat3 signaling pathway by nifuroxazide improves antitumor immunity and impairs colorectal carcinoma metastasis. [electronic resource] by
- Ye, Ting-Hong
- Yang, Fang-Fang
- Zhu, Yong-Xia
- Li, Ya-Li
- Lei, Qian
- Song, Xue-Jiao
- Xia, Yong
- Xiong, Ying
- Zhang, Li-Dan
- Wang, Ning-Yu
- Zhao, Li-Feng
- Gou, Hong-Feng
- Xie, Yong-Mei
- Yang, Sheng-Yong
- Yu, Luo-Ting
- Yang, Li
- Wei, Yu-Quan
Publication details: Cell death & disease Sep 2019
In:
Cell death & disease vol. 10
Availability: No items available.
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116.
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Design, Synthesis, and Structure-Activity Relationship Studies of 3-(Phenylethynyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine Derivatives as a New Class of Src Inhibitors with Potent Activities in Models of Triple Negative Breast Cancer. [electronic resource] by
- Zhang, Chun-Hui
- Zheng, Ming-Wu
- Li, Ya-Ping
- Lin, Xing-Dong
- Huang, Mei
- Zhong, Lei
- Li, Guo-Bo
- Zhang, Rong-Jie
- Lin, Wan-Ting
- Jiao, Yan
- Wu, Xiao-Ai
- Yang, Jiao
- Xiang, Rong
- Chen, Li-Juan
- Zhao, Ying-Lan
- Cheng, Wei
- Wei, Yu-Quan
- Yang, Sheng-Yong
Producer: 20150806
In:
Journal of medicinal chemistry vol. 58
Availability: No items available.
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117.
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From Lead to Drug Candidate: Optimization of 3-(Phenylethynyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine Derivatives as Agents for the Treatment of Triple Negative Breast Cancer. [electronic resource] by
- Zhang, Chun-Hui
- Chen, Kai
- Jiao, Yan
- Li, Lin-Li
- Li, Ya-Ping
- Zhang, Rong-Jie
- Zheng, Ming-Wu
- Zhong, Lei
- Huang, Shen-Zhen
- Song, Chun-Li
- Lin, Wan-Ting
- Yang, Jiao
- Xiang, Rong
- Peng, Bing
- Han, Jun-Hong
- Lu, Guang-Wen
- Wei, Yu-Quan
- Yang, Sheng-Yong
Producer: 20170608
In:
Journal of medicinal chemistry vol. 59
Availability: No items available.
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118.
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Discovery of the novel potent and selective FLT3 inhibitor 1-{5-[7-(3- morpholinopropoxy)quinazolin-4-ylthio]-[1,3,4]thiadiazol-2-yl}-3-p-tolylurea and its anti-acute myeloid leukemia (AML) activities in vitro and in vivo. [electronic resource] by
- Li, Wei-Wei
- Wang, Xiao-Yan
- Zheng, Ren-Lin
- Yan, Heng-Xiu
- Cao, Zhi-Xing
- Zhong, Lei
- Wang, Ze-Rong
- Ji, Pan
- Yang, Ling-Ling
- Wang, Li-Jiao
- Xu, Yong
- Liu, Jing-Jing
- Yang, Jiao
- Zhang, Chun-Hui
- Ma, Shuang
- Feng, Shan
- Sun, Qi-Zheng
- Wei, Yu-Quan
- Yang, Sheng-Yong
Producer: 20120717
In:
Journal of medicinal chemistry vol. 55
Availability: No items available.
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119.
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Discovery of imidazo[2,1-b]thiazole HCV NS4B inhibitors exhibiting synergistic effect with other direct-acting antiviral agents. [electronic resource] by
- Wang, Ning-Yu
- Xu, Ying
- Zuo, Wei-Qiong
- Xiao, Kun-Jie
- Liu, Li
- Zeng, Xiu-Xiu
- You, Xin-Yu
- Zhang, Li-Dan
- Gao, Chao
- Liu, Zhi-Hao
- Ye, Ting-Hong
- Xia, Yong
- Xiong, Ying
- Song, Xue-Jiao
- Lei, Qian
- Peng, Cui-Ting
- Tang, Hong
- Yang, Sheng-Yong
- Wei, Yu-Quan
- Yu, Luo-Ting
Producer: 20150526
In:
Journal of medicinal chemistry vol. 58
Availability: No items available.
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