Carroll, C D

Identification of potent inhibitors of Plasmodium falciparum plasmepsin II from an encoded statine combinatorial library. [electronic resource] - Bioorganic & medicinal chemistry letters Sep 1998 - 2315-20 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

0960-894X

10.1016/s0960-894x(98)00419-3 doi


Amino Acids
Animals
Antimalarials--chemical synthesis
Aspartic Acid Endopeptidases--antagonists & inhibitors
Cloning, Molecular
Databases as Topic
Drug Design
Hemoglobins--metabolism
Humans
Molecular Structure
Oligopeptides--chemical synthesis
Peptide Library
Plasmodium falciparum--enzymology
Protease Inhibitors--chemical synthesis
Protozoan Proteins
Recombinant Proteins--antagonists & inhibitors
Structure-Activity Relationship
Substrate Specificity