Fry, D W

Specific, irreversible inactivation of the epidermal growth factor receptor and erbB2, by a new class of tyrosine kinase inhibitor. [electronic resource] - Proceedings of the National Academy of Sciences of the United States of America Sep 1998 - 12022-7 p. digital

Publication Type: Journal Article

0027-8424

10.1073/pnas.95.20.12022 doi


Animals
Antineoplastic Agents--chemistry
Binding Sites--genetics
Cell Line
Cysteine--chemistry
Enzyme Inhibitors--chemistry
ErbB Receptors--antagonists & inhibitors
Humans
Mice
Mice, Nude
Models, Molecular
Mutagenesis, Site-Directed
Neoplasm Transplantation
Neoplasms, Experimental--drug therapy
Protein Conformation
Protein-Tyrosine Kinases--antagonists & inhibitors
Quinazolines--chemistry
Receptor, ErbB-2--antagonists & inhibitors
Recombinant Fusion Proteins--antagonists & inhibitors
Transplantation, Heterologous
Tumor Cells, Cultured