Chimirri, A 3,5-Dihydro-4H-2,3-benzodiazepine-4-thiones: a new class of AMPA receptor antagonists. [electronic resource] - Journal of medicinal chemistry Aug 1998 - 3409-16 p. digital Publication Type: Journal Article; Research Support, Non-U.S. Gov't ISSN: 0022-2623 Standard No.: 10.1021/jm9800393 doi Subjects--Topical Terms: Acoustic StimulationAnimalsAnticonvulsants--chemical synthesisBenzodiazepines--chemical synthesisConvulsants--toxicityElectroshockExcitatory Amino Acid Agonists--toxicityExcitatory Amino Acid Antagonists--chemical synthesisGuinea PigsIn Vitro TechniquesMaleMiceMice, Inbred DBAMotor Activity--drug effectsOlfactory Pathways--drug effectsPatch-Clamp TechniquesPentylenetetrazole--toxicityPyrrolidinones--pharmacologyRatsReceptors, AMPA--antagonists & inhibitorsSeizures--drug therapyStructure-Activity RelationshipThiones--chemical synthesisalpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid--toxicity