Kudo, S

Involvement of human cytochrome P450 3A4 in reduced haloperidol oxidation. [electronic resource] - European journal of clinical pharmacology May 1998 - 253-9 p. digital

Publication Type: Journal Article

0031-6970

10.1007/s002280050455 doi


Anti-Arrhythmia Agents--pharmacology
Anti-Bacterial Agents--administration & dosage
Antiparkinson Agents--pharmacology
Biotransformation--drug effects
Biperiden--pharmacology
Carteolol--metabolism
Cell Line, Transformed
Cytochrome P-450 CYP2D6--metabolism
Cytochrome P-450 CYP2D6 Inhibitors
Cytochrome P-450 CYP3A
Cytochrome P-450 Enzyme Inhibitors
Cytochrome P-450 Enzyme System--metabolism
Dose-Response Relationship, Drug
Haloperidol--antagonists & inhibitors
Humans
Hydroxylation--drug effects
Isoenzymes--antagonists & inhibitors
Kinetics
Microsomes--drug effects
Mixed Function Oxygenases--antagonists & inhibitors
Oxidation-Reduction--drug effects
Quinidine--pharmacology
Sparteine--pharmacology
Troleandomycin--administration & dosage