Boger, D L

Design, synthesis, and evaluation of potential GAR and AICAR transformylase inhibitors. [electronic resource] - Bioorganic & medicinal chemistry Jun 1998 - 643-59 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't; Research Support, U.S. Gov't, P.H.S.

0968-0896

10.1016/s0968-0896(98)00040-6 doi


Animals
Antineoplastic Agents--chemical synthesis
Drug Design
Drug Screening Assays, Antitumor
Enzyme Inhibitors--chemical synthesis
Hydroxymethyl and Formyl Transferases--antagonists & inhibitors
Mice
Phosphoribosylaminoimidazolecarboxamide Formyltransferase
Phosphoribosylglycinamide Formyltransferase
Pyrimidines--chemical synthesis
Quinazolines--chemical synthesis
Structure-Activity Relationship
Tumor Cells, Cultured