TY  - GEN
AU  - Albright,J D
AU  - Reich,M F
AU  - Delos Santos,E G
AU  - Dusza,J P
AU  - Sum,F W
AU  - Venkatesan,A M
AU  - Coupet,J
AU  - Chan,P S
AU  - Ru,X
AU  - Mazandarani,H
AU  - Bailey,T
TI  - 5-Fluoro-2-methyl-N-[4-(5H-pyrrolo[2,1-c]-[1, 4]benzodiazepin-10(11H)-ylcarbonyl)-3-chlorophenyl]benzamide (VPA-985): an orally active arginine vasopressin antagonist with selectivity for V2 receptors
SN  - 0022-2623
PY  - 1998///0724
KW  - Administration, Oral
KW  - Animals
KW  - Arginine Vasopressin
KW  - antagonists & inhibitors
KW  - Azepines
KW  - administration & dosage
KW  - Benzamides
KW  - Blood Platelets
KW  - metabolism
KW  - Body Water
KW  - Cell Line
KW  - Cell Membrane
KW  - Dogs
KW  - Fibroblasts
KW  - drug effects
KW  - Humans
KW  - Kidney
KW  - Liver
KW  - Osmolar Concentration
KW  - Pyrroles
KW  - Rats
KW  - Receptors, Vasopressin
KW  - Sodium
KW  - blood
KW  - Structure-Activity Relationship
KW  - Urine
KW  - chemistry
N1  - Publication Type: Clinical Trial; Journal Article; Randomized Controlled Trial
UR  - https://doi.org/10.1021/jm980179c
ER  -