Szardenings, A K Rational design and combinatorial evaluation of enzyme inhibitor scaffolds: identification of novel inhibitors of matrix metalloproteinases. [electronic resource] - Journal of medicinal chemistry Jun 1998 - 2194-200 p. digital Publication Type: Journal Article ISSN: 0022-2623 Standard No.: 10.1021/jm980133j doi Subjects--Topical Terms: DiketopiperazinesDrug DesignEnzyme Inhibitors--chemical synthesisHumansHydrogen BondingMatrix Metalloproteinase 1Matrix Metalloproteinase 9Matrix Metalloproteinase InhibitorsMetalloendopeptidases--antagonists & inhibitorsPiperazines--chemical synthesisStructure-Activity Relationship