Egorin, M J

Metabolism of 17-(allylamino)-17-demethoxygeldanamycin (NSC 330507) by murine and human hepatic preparations. [electronic resource] - Cancer research Jun 1998 - 2385-96 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't; Research Support, U.S. Gov't, P.H.S.

0008-5472


Animals
Antibiotics, Antineoplastic--metabolism
Benzoquinones
Cells, Cultured
Chromatography, High Pressure Liquid
Cytochrome P-450 CYP3A
Cytochrome P-450 Enzyme System--metabolism
Cytosol--drug effects
Epoxide Hydrolases--metabolism
Gas Chromatography-Mass Spectrometry
Humans
Ketoconazole--pharmacology
Lactams, Macrocyclic
Liver--drug effects
Mice
Microsomes, Liver--drug effects
Mixed Function Oxygenases--metabolism
Molecular Weight
NAD--metabolism
Quinones--metabolism
Rifabutin--analogs & derivatives
Species Specificity