Pälvimäki, E P

Deramciclane, a putative anxiolytic drug, is a serotonin 5-HT2C receptor inverse agonist but fails to induce 5-HT2C receptor down-regulation. [electronic resource] - Psychopharmacology Mar 1998 - 99-104 p. digital

Publication Type: Comparative Study; Journal Article; Research Support, Non-U.S. Gov't

0033-3158

10.1007/s002130050544 doi


Animals
Anti-Anxiety Agents--pharmacology
Brain--drug effects
Camphanes--pharmacology
Clozapine--pharmacology
Inositol Phosphates--metabolism
Male
Rats
Rats, Sprague-Dawley
Receptor, Serotonin, 5-HT2A
Receptor, Serotonin, 5-HT2C
Receptors, Serotonin--drug effects
Serotonin Antagonists--pharmacology