Barr, A J

Agonist-independent activation of Gz by the 5-hydroxytryptamine1A receptor co-expressed in Spodoptera frugiperda cells. Distinguishing inverse agonists from neutral antagonists. [electronic resource] - The Journal of biological chemistry Dec 1997 - 32979-87 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't; Research Support, U.S. Gov't, P.H.S.

0021-9258

10.1074/jbc.272.52.32979 doi


Aminopyridines--metabolism
Animals
Enzyme Inhibitors--metabolism
GTP-Binding Protein alpha Subunits
GTP-Binding Proteins--metabolism
Guanosine 5'-O-(3-Thiotriphosphate)--metabolism
Heterotrimeric GTP-Binding Proteins
Humans
Kinetics
Ligands
Piperazines--metabolism
Receptors, Serotonin--metabolism
Receptors, Serotonin, 5-HT1
Serotonin Antagonists--metabolism
Spiperone--metabolism
Spodoptera
Tetrahydronaphthalenes--metabolism