Li, A P

Primary human hepatocytes as a tool for the evaluation of structure-activity relationship in cytochrome P450 induction potential of xenobiotics: evaluation of rifampin, rifapentine and rifabutin. [electronic resource] - Chemico-biological interactions Nov 1997 - 17-30 p. digital

Publication Type: Comparative Study; Journal Article

0009-2797

10.1016/s0009-2797(97)00071-9 doi


Antibiotics, Antitubercular--metabolism
Antitubercular Agents--metabolism
Cytochrome P-450 Enzyme System--biosynthesis
Drug Evaluation, Preclinical--methods
Enzyme Induction--drug effects
Glucuronates--metabolism
Humans
Hydroxylation
Isoenzymes--biosynthesis
Liver--cytology
Rifabutin--metabolism
Rifampin--analogs & derivatives
Structure-Activity Relationship
Testosterone--metabolism
Time Factors
Zidovudine--metabolism