Feng, D M

Discovery of a novel, selective, and orally bioavailable class of thrombin inhibitors incorporating aminopyridyl moieties at the P1 position. [electronic resource] - Journal of medicinal chemistry Nov 1997 - 3726-33 p. digital

Publication Type: Journal Article

0022-2623

10.1021/jm970493r doi


Administration, Oral
Animals
Antithrombins--chemical synthesis
Biological Availability
Crystallography, X-Ray
Dipeptides--chemical synthesis
Dogs
Kinetics
Pyridines--chemical synthesis
Rats
Structure-Activity Relationship
Thrombin--antagonists & inhibitors