Ren, S

Oxidation of cyclophosphamide to 4-hydroxycyclophosphamide and deschloroethylcyclophosphamide in human liver microsomes. [electronic resource] - Cancer research Oct 1997 - 4229-35 p. digital

Publication Type: Comparative Study; Journal Article; Research Support, U.S. Gov't, P.H.S.

0008-5472


Aryl Hydrocarbon Hydroxylases
Biotransformation
Cyclophosphamide--analogs & derivatives
Cytochrome P-450 CYP2C9
Cytochrome P-450 CYP3A
Cytochrome P-450 Enzyme Inhibitors
Cytochrome P-450 Enzyme System--genetics
Enzyme Inhibitors--pharmacology
Humans
Isoenzymes--antagonists & inhibitors
Kinetics
Microsomes, Liver--metabolism
Mixed Function Oxygenases--antagonists & inhibitors
Orphenadrine--pharmacology
Oxidation-Reduction
Prodrugs--metabolism
Recombinant Fusion Proteins--metabolism
Steroid 16-alpha-Hydroxylase
Steroid Hydroxylases--antagonists & inhibitors
Troleandomycin--pharmacology