Mechanism of action of fotemustine, a new chloroethylnitrosourea anticancer agent: evidence for the formation of two DNA-reactive intermediates contributing to cytotoxicity. [electronic resource]
- Biochemistry Sep 1997
- 10646-54 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
0006-2960
10.1021/bi970791q doi
Antineoplastic Agents--metabolism Cell Survival--drug effects DNA Adducts--metabolism DNA Methylation--drug effects DNA Repair--drug effects Dose-Response Relationship, Drug Drug Stability Guanine--metabolism HeLa Cells Humans Mass Spectrometry Melanoma Nitrosourea Compounds--metabolism Organophosphorus Compounds--metabolism Tumor Cells, Cultured