TY  - GEN
AU  - Giardina,G A
AU  - Sarau,H M
AU  - Farina,C
AU  - Medhurst,A D
AU  - Grugni,M
AU  - Raveglia,L F
AU  - Schmidt,D B
AU  - Rigolio,R
AU  - Luttmann,M
AU  - Vecchietti,V
AU  - Hay,D W
TI  - Discovery of a novel class of selective non-peptide antagonists for the human neurokinin-3 receptor. 1. Identification of the 4-quinolinecarboxamide framework
SN  - 0022-2623
PY  - 1997///0715
KW  - Animals
KW  - Binding, Competitive
KW  - CHO Cells
KW  - Chemical Phenomena
KW  - Chemistry, Physical
KW  - Cricetinae
KW  - Humans
KW  - Hydrogen Bonding
KW  - Molecular Structure
KW  - Muscle Contraction
KW  - drug effects
KW  - Peptide Fragments
KW  - pharmacology
KW  - Quinolines
KW  - chemical synthesis
KW  - Rabbits
KW  - Receptors, Neurokinin-3
KW  - antagonists & inhibitors
KW  - Recombinant Proteins
KW  - metabolism
KW  - Stereoisomerism
KW  - Structure-Activity Relationship
KW  - Substance P
KW  - analogs & derivatives
N1  - Publication Type: Journal Article
UR  - https://doi.org/10.1021/jm960818o
ER  -