Giardina, G A <br/><br/>
Discovery of a novel class of selective non-peptide antagonists for the human neurokinin-3 receptor. 1. Identification of the 4-quinolinecarboxamide framework.  [electronic resource] 

 -  Journal of medicinal chemistry  Jun 1997 
 - 1794-807 p.  digital 
<br/><br/> Publication Type: Journal Article 
<br/><br/><label>ISSN: </label>0022-2623 
<br/><br/><label>Standard No.: </label>10.1021/jm960818o  doi 
<br/><br/><label>Subjects--Topical Terms: </label><br/>Animals<br/>Binding, Competitive<br/>CHO Cells<br/>Chemical Phenomena<br/>Chemistry, Physical<br/>Cricetinae<br/>Humans<br/>Hydrogen Bonding<br/>Molecular Structure<br/>Muscle Contraction--drug effects<br/>Peptide Fragments--pharmacology<br/>Quinolines--chemical synthesis<br/>Rabbits<br/>Receptors, Neurokinin-3--antagonists & inhibitors<br/>Recombinant Proteins--metabolism<br/>Stereoisomerism<br/>Structure-Activity Relationship<br/>Substance P--analogs & derivatives