Biologically active conformer of the effector region of human C5a and modulatory effects of N-terminal receptor binding determinants on activity. [electronic resource]
- Journal of medicinal chemistry Mar 1997
- 877-84 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
0022-2623
10.1021/jm960727r doi
Antigens, CD--metabolism Arteries--drug effects Binding, Competitive Complement C5a--agonists Fetus Glucuronidase--metabolism Humans In Vitro Techniques Muscle, Smooth, Vascular--drug effects Neutrophils--drug effects Peptide Fragments--chemistry Protein Binding Protein Conformation Protein Structure, Secondary Receptor, Anaphylatoxin C5a Receptors, Complement--metabolism Vasoconstriction--drug effects