Reversal of P-glycoprotein is greatly reduced by the presence of plasma but can be monitored by an ex vivo clinical assay. [electronic resource]
- Anti-cancer drugs Aug 1996
- 678-86 p. digital
Publication Type: Comparative Study; Journal Article; Research Support, Non-U.S. Gov't; Research Support, U.S. Gov't, Non-P.H.S.
0959-4973
10.1097/00001813-199608000-00009 doi
ATP Binding Cassette Transporter, Subfamily B, Member 1--antagonists & inhibitors Animals Cyclosporine--blood Daunorubicin--metabolism Drug Screening Assays, Antitumor Humans Kidney--metabolism Leukemia P388--drug therapy Mice Plasma Quinidine--blood Verapamil--pharmacology Vinblastine--metabolism