Feierman, D E

Metabolism of fentanyl, a synthetic opioid analgesic, by human liver microsomes. Role of CYP3A4. [electronic resource] - Drug metabolism and disposition: the biological fate of chemicals Sep 1996 - 932-9 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't; Research Support, U.S. Gov't, P.H.S.

0090-9556


Analgesics, Opioid--metabolism
Aryl Hydrocarbon Hydroxylases
Cytochrome P-450 CYP1A2--metabolism
Cytochrome P-450 CYP2C8
Cytochrome P-450 CYP2C9
Cytochrome P-450 CYP3A
Cytochrome P-450 Enzyme Inhibitors
Cytochrome P-450 Enzyme System--metabolism
Fentanyl--analogs & derivatives
Gas Chromatography-Mass Spectrometry
Humans
Ketoconazole--pharmacology
Kinetics
Microsomes, Liver--enzymology
Mixed Function Oxygenases--antagonists & inhibitors
Steroid 16-alpha-Hydroxylase
Steroid Hydroxylases--metabolism
Theophylline--analogs & derivatives
Tolbutamide--pharmacology