GR205171: a novel antagonist with high affinity for the tachykinin NK1 receptor, and potent broad-spectrum anti-emetic activity. [electronic resource]
- Regulatory peptides Aug 1996
- 45-53 p. digital
Publication Type: Journal Article
0167-0115
10.1016/0167-0115(96)00071-7 doi
Administration, Oral Animals Antiemetics--metabolism Cisplatin--adverse effects Dogs Dose-Response Relationship, Drug Ferrets Humans Male Motor Activity Neurokinin-1 Receptor Antagonists Piperidines--metabolism Receptors, Neurokinin-1--metabolism Shrews Stereoisomerism Tetrazoles--metabolism