TY  - GEN
AU  - Campiani,G
AU  - Fiorini,I
AU  - De Filippis,M P
AU  - Ciani,S M
AU  - Garofalo,A
AU  - Nacci,V
AU  - Giorgi,G
AU  - Sega,A
AU  - Botta,M
AU  - Chiarini,A
AU  - Budriesi,R
AU  - Bruni,G
AU  - Romeo,M R
AU  - Manzoni,C
AU  - Mennini,T
TI  - Cardiovascular characterization of pyrrolo[2,1-d][1,5]benzothiazepine derivatives binding selectively to the peripheral-type benzodiazepine receptor (PBR): from dual PBR affinity and calcium antagonist activity to novel and selective calcium entry blockers
SN  - 0022-2623
PY  - 1996///0906
KW  - Animals
KW  - Atrial Function
KW  - Binding, Competitive
KW  - Calcium Channel Blockers
KW  - chemical synthesis
KW  - Calcium Channels
KW  - metabolism
KW  - Cardiovascular System
KW  - drug effects
KW  - Cerebral Cortex
KW  - Depression, Chemical
KW  - Female
KW  - Guinea Pigs
KW  - Heart Rate
KW  - Male
KW  - Models, Molecular
KW  - Myocardial Contraction
KW  - Myocardium
KW  - Pyrroles
KW  - Rats
KW  - Rats, Sprague-Dawley
KW  - Receptors, GABA-A
KW  - Structure-Activity Relationship
KW  - Thiazepines
N1  - Publication Type: Comparative Study; Journal Article; Research Support, Non-U.S. Gov't
UR  - https://doi.org/10.1021/jm960162z
ER  -