Ladduwahetty, T N-heteroaryl-2-phenyl-3-(benzyloxy)piperidines: a novel class of potent orally active human NK1 antagonists. [electronic resource] - Journal of medicinal chemistry Jul 1996 - 2907-14 p. digital Publication Type: Journal Article ISSN: 0022-2623 Standard No.: 10.1021/jm9506534 doi Subjects--Topical Terms: AnimalsBiological AvailabilityDrug StabilityFerretsGuinea PigsHumansInflammation--drug therapyMacaca mulattaMaleMicrosomes, Liver--metabolismMigraine Disorders--drug therapyNeurokinin-1 Receptor AntagonistsPiperidines--chemical synthesisRatsReceptors, Neurokinin-1--metabolismTriazoles--chemical synthesisVomiting--drug therapy