Stable guanosine 5'-triphosphate-analogues inhibit specific (+)-[3H]isradipine binding in rat hearts by a Ca(2+)-lowering, G protein-independent mechanism. [electronic resource]
- Pharmacology & toxicology Jan 1996
- 28-36 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
0901-9928
10.1111/j.1600-0773.1996.tb00176.x doi
Animals Calcium--metabolism Calcium Channels--drug effects Cyclic AMP-Dependent Protein Kinases--metabolism GTP-Binding Proteins--metabolism Guanosine 5'-O-(3-Thiotriphosphate)--pharmacology Guanylyl Imidodiphosphate--pharmacology Heart--drug effects In Vitro Techniques Isradipine--pharmacokinetics Magnesium--pharmacology Male Membranes--drug effects Myocardium--cytology Radioligand Assay Rats Rats, Wistar Temperature Vasodilator Agents--pharmacokinetics