Williams, D L Pharmacology of L-754,142, a highly potent, orally active, nonpeptidyl endothelin antagonist. [electronic resource] - The Journal of pharmacology and experimental therapeutics Dec 1995 - 1518-26 p. digital Publication Type: Journal Article ISSN: 0022-3565 Subjects--Topical Terms: Acetamides--pharmacokineticsAdministration, OralAnimalsBiological AvailabilityBlood Pressure--drug effectsCHO CellsCricetinaeEndothelin Receptor AntagonistsEndothelins--antagonists & inhibitorsFerretsHumansHydrolysisIn Vitro TechniquesMaleMiceMuscle Contraction--drug effectsMuscle, Smooth, Vascular--drug effectsPhosphatidylinositols--metabolismRabbitsRatsRats, Sprague-DawleyReceptors, Endothelin--metabolism