Paul, R Preparation of substituted N-phenyl-4-aryl-2-pyrimidinamines as mediator release inhibitors. [electronic resource] - Journal of medicinal chemistry Sep 1993 - 2716-25 p. digital Publication Type: Journal Article ISSN: 0022-2623 Standard No.: 10.1021/jm00071a002 doi Subjects--Topical Terms: AnimalsBasophils--drug effectsFemaleHistamine Antagonists--chemical synthesisHumansImidazoles--chemical synthesisLethal Dose 50Macaca mulattaMaleMicePassive Cutaneous Anaphylaxis--drug effectsPyrimidines--chemical synthesisRatsRats, Sprague-DawleyStructure-Activity Relationship