Sanghani, P C

A strategy for the design of membrane-permeable folypoly-gamma-glutamate synthetase inhibitors: "bay-region"-substituted 2-desamino-2-methyl-5,8-dideazafolate analogs. [electronic resource] - Molecular pharmacology Feb 1994 - 341-51 p. digital

Publication Type: Journal Article; Research Support, U.S. Gov't, P.H.S.

0026-895X


Animals
Binding Sites
Cell Division--drug effects
Cell Membrane Permeability
Drug Design
Female
Folic Acid--analogs & derivatives
Mice
Peptide Synthases--antagonists & inhibitors
Structure-Activity Relationship
Tumor Cells, Cultured