Murray, M

Competitive inhibition of human liver microsomal cytochrome P450 3A-dependent steroid 6 beta-hydroxylation activity by cyclophosphamide and ifosfamide in vitro. [electronic resource] - The Journal of pharmacology and experimental therapeutics Aug 1994 - 645-9 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

0022-3565


Acrolein--metabolism
Animals
Binding, Competitive
Cyclophosphamide--pharmacology
Cytochrome P-450 CYP2E1
Cytochrome P-450 Enzyme Inhibitors
Cytochrome P-450 Enzyme System--metabolism
Humans
Ifosfamide--pharmacology
Microsomes, Liver--drug effects
Mixed Function Oxygenases--antagonists & inhibitors
NADP--metabolism
Rats
Rats, Wistar
Steroid Hydroxylases--metabolism
Testosterone--metabolism