Modification by brefeldin A, bafilomycin A1 and 7-chloro-4-nitrobenz-2-oxa-1,3-diazole (NBD) of cellular accumulation and intracellular distribution of anthracyclines in the non-P-glycoprotein-mediated multidrug-resistant cell line COR-L23/R. [electronic resource]
- British journal of cancer Jul 1994
- 60-6 p. digital
Publication Type: Journal Article
0007-0920
10.1038/bjc.1994.250 doi
4-Chloro-7-nitrobenzofurazan--pharmacology ATP Binding Cassette Transporter, Subfamily B, Member 1 Anti-Bacterial Agents--pharmacology Antibiotics, Antineoplastic--pharmacokinetics Brefeldin A Carcinoma, Non-Small-Cell Lung--metabolism Carrier Proteins Cell Nucleus--metabolism Cyclopentanes--pharmacology Cytoplasm--metabolism Daunorubicin--pharmacokinetics Doxorubicin--pharmacokinetics Drug Interactions Drug Resistance--physiology Drug Screening Assays, Antitumor Golgi Apparatus--drug effects Humans Lung Neoplasms--metabolism Macrolides Membrane Glycoproteins Protein Synthesis Inhibitors--pharmacology Proton-Translocating ATPases--antagonists & inhibitors Tetrazolium Salts Thiazoles Tumor Cells, Cultured--drug effects