Hancock, A A

Preclinical pharmacological actions of (+/-)-(1'R*,3R*)-3-phenyl-1- [1',2',3',4'-tetrahydro-5',6'-methylene-dioxy-1'-naphthalenyl) methyl] pyrrolidine methanesulfonate (ABT-200), a potential antidepressant agent that antagonizes alpha-2 adrenergic receptors and inhibits the neuronal uptake of norepinephrine. [electronic resource] - The Journal of pharmacology and experimental therapeutics Mar 1995 - 1160-9 p. digital

Publication Type: Journal Article

0022-3565


Adrenergic Uptake Inhibitors--pharmacology
Adrenergic alpha-2 Receptor Antagonists
Animals
Antidepressive Agents--pharmacology
Behavior, Animal--drug effects
Blood Pressure--drug effects
Clonidine--pharmacology
Guinea Pigs
Heart Rate--drug effects
Hippocampus--metabolism
In Vitro Techniques
Male
Motor Activity--drug effects
Mydriasis--chemically induced
Neurons--metabolism
Olfactory Bulb--physiology
Pyrrolidines--pharmacology
Rabbits
Radioligand Assay
Rats
Rats, Sprague-Dawley
Synaptosomes--metabolism
Tyramine--analogs & derivatives