TY - GEN AU - Hlasta,D J AU - Subramanyam,C AU - Bell,M R AU - Carabateas,P M AU - Court,J J AU - Desai,R C AU - Drozd,M L AU - Eickhoff,W M AU - Ferguson,E W AU - Gordon,R J TI - Orally bioavailable benzisothiazolone inhibitors of human leukocyte elastase SN - 0022-2623 PY - 1995///0404 KW - Administration, Oral KW - Animals KW - Biological Availability KW - Chlorobenzoates KW - chemical synthesis KW - Cricetinae KW - Dogs KW - Drug Stability KW - Humans KW - In Vitro Techniques KW - Leukocyte Elastase KW - Lung KW - enzymology KW - Macaca fascicularis KW - Mesocricetus KW - Pancreatic Elastase KW - antagonists & inhibitors KW - Rats KW - Rats, Sprague-Dawley KW - Thiazoles N1 - Publication Type: Journal Article UR - https://doi.org/10.1021/jm00005a001 ER -