Hlasta, D J Orally bioavailable benzisothiazolone inhibitors of human leukocyte elastase. [electronic resource] - Journal of medicinal chemistry Mar 1995 - 739-44 p. digital Publication Type: Journal Article ISSN: 0022-2623 Standard No.: 10.1021/jm00005a001 doi Subjects--Topical Terms: Administration, OralAnimalsBiological AvailabilityChlorobenzoates--chemical synthesisCricetinaeDogsDrug StabilityHumansIn Vitro TechniquesLeukocyte ElastaseLung--enzymologyMacaca fascicularisMesocricetusPancreatic Elastase--antagonists & inhibitorsRatsRats, Sprague-DawleyThiazoles--chemical synthesis