Hlasta, D J

Orally bioavailable benzisothiazolone inhibitors of human leukocyte elastase. [electronic resource] - Journal of medicinal chemistry Mar 1995 - 739-44 p. digital

Publication Type: Journal Article

0022-2623

10.1021/jm00005a001 doi


Administration, Oral
Animals
Biological Availability
Chlorobenzoates--chemical synthesis
Cricetinae
Dogs
Drug Stability
Humans
In Vitro Techniques
Leukocyte Elastase
Lung--enzymology
Macaca fascicularis
Mesocricetus
Pancreatic Elastase--antagonists & inhibitors
Rats
Rats, Sprague-Dawley
Thiazoles--chemical synthesis