Functional analysis of P-glycoprotein mutants identifies predicted transmembrane domain 11 as a putative drug binding site. [electronic resource]
- Biochemistry Apr 1993
- 4185-94 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't; Research Support, U.S. Gov't, P.H.S.
0006-2960
10.1021/bi00067a005 doi
ATP Binding Cassette Transporter, Subfamily B, Member 1 Affinity Labels Amino Acid Sequence Animals Azides--metabolism Binding Sites Biological Transport CHO Cells Cell Membrane--metabolism Cloning, Molecular Colchicine--metabolism Cricetinae Dactinomycin--metabolism Doxorubicin Drug Resistance--genetics Gramicidin--metabolism Iodine Radioisotopes Kinetics Membrane Glycoproteins--genetics Mice Mutagenesis, Site-Directed Phenylalanine Prazosin--analogs & derivatives Serine Transfection Vinblastine--metabolism