Bétoin, F

In vitro and in vivo evidence for a tachykinin NK1 receptor antagonist effect of vapreotide, an analgesic cyclic analog of somatostatin. [electronic resource] - European journal of pharmacology Jun 1995 - 241-9 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

0014-2999

10.1016/0014-2999(95)00168-k doi


Acetylcholine--pharmacology
Analgesics--metabolism
Animals
Binding, Competitive--drug effects
Brain--metabolism
Bronchi--drug effects
Capillary Permeability--drug effects
Duodenum--drug effects
Electric Stimulation
Female
Guinea Pigs
In Vitro Techniques
Injections, Spinal
Male
Mice
Muscle Contraction--drug effects
Muscle, Smooth--drug effects
Neurokinin A--analogs & derivatives
Neurokinin-1 Receptor Antagonists
Peptide Fragments--pharmacology
Rats
Rats, Sprague-Dawley
Receptors, Neurokinin-1--metabolism
Somatostatin--analogs & derivatives
Substance P--metabolism