Sayre, L M

Design and synthesis of naltrexone-derived affinity labels with nonequilibrium opioid agonist and antagonist activities. Evidence for the existence of different mu receptor subtypes in different tissues. [electronic resource] - Journal of medicinal chemistry Oct 1984 - 1325-35 p. digital

Publication Type: Comparative Study; Journal Article; Research Support, U.S. Gov't, P.H.S.

0022-2623

10.1021/jm00376a018 doi


Affinity Labels--chemical synthesis
Animals
Chemical Phenomena
Chemistry
Guinea Pigs
Ileum--drug effects
Indicators and Reagents
Kinetics
Magnetic Resonance Spectroscopy
Male
Mice
Morphine--pharmacology
Muscle, Smooth--drug effects
Naloxone--analogs & derivatives
Naltrexone--analogs & derivatives
Receptors, Opioid--drug effects
Receptors, Opioid, mu
Structure-Activity Relationship
Vas Deferens--drug effects