Bock, M G Cholecystokinin antagonists. Synthesis of asperlicin analogues with improved potency and water solubility. [electronic resource] - Journal of medicinal chemistry Oct 1986 - 1941-5 p. digital Publication Type: Journal Article ISSN: 0022-2623 Standard No.: 10.1021/jm00160a024 doi Subjects--Topical Terms: AnimalsBenzodiazepinones--chemical synthesisCholecystokinin--antagonists & inhibitorsGuinea PigsIn Vitro TechniquesRatsReceptors, Cholecystokinin--drug effectsSolubilityStructure-Activity Relationship