A phase I evaluation of the quinazoline antifolate thymidylate synthase inhibitor, N10-propargyl-5,8-dideazafolic acid, CB3717. [electronic resource]
- Journal of clinical oncology : official journal of the American Society of Clinical Oncology Aug 1986
- 1245-52 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
0732-183X
10.1200/JCO.1986.4.8.1245 doi
Acetylglucosaminidase--urine Acid Phosphatase--blood Alanine Transaminase--blood Antineoplastic Agents--administration & dosage Chemical and Drug Induced Liver Injury Dose-Response Relationship, Drug Drug Administration Schedule Drug Evaluation Folic Acid--analogs & derivatives Folic Acid Antagonists--administration & dosage Glomerular Filtration Rate--drug effects Hematologic Diseases--chemically induced Hyperbilirubinemia--chemically induced Kidney Diseases--chemically induced Leucyl Aminopeptidase--urine Neoplasms--blood Quinazolines--administration & dosage Skin Diseases--chemically induced Thymidylate Synthase--antagonists & inhibitors