Calvert, A H

A phase I evaluation of the quinazoline antifolate thymidylate synthase inhibitor, N10-propargyl-5,8-dideazafolic acid, CB3717. [electronic resource] - Journal of clinical oncology : official journal of the American Society of Clinical Oncology Aug 1986 - 1245-52 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

0732-183X

10.1200/JCO.1986.4.8.1245 doi


Acetylglucosaminidase--urine
Acid Phosphatase--blood
Alanine Transaminase--blood
Antineoplastic Agents--administration & dosage
Chemical and Drug Induced Liver Injury
Dose-Response Relationship, Drug
Drug Administration Schedule
Drug Evaluation
Folic Acid--analogs & derivatives
Folic Acid Antagonists--administration & dosage
Glomerular Filtration Rate--drug effects
Hematologic Diseases--chemically induced
Hyperbilirubinemia--chemically induced
Kidney Diseases--chemically induced
Leucyl Aminopeptidase--urine
Neoplasms--blood
Quinazolines--administration & dosage
Skin Diseases--chemically induced
Thymidylate Synthase--antagonists & inhibitors