Stein, R L Mechanism for slow-binding inhibition of human leukocyte elastase by valine-derived benzoxazinones. [electronic resource] - Biochemistry Jun 1987 - 4126-30 p. digital Publication Type: Journal Article ISSN: 0006-2960 Standard No.: 10.1021/bi00387a057 doi Subjects--Topical Terms: AcylationBinding Sites--drug effectsBinding, CompetitiveEnzyme Inhibitors--pharmacologyHumansKineticsLeukocytes--enzymologyOxazines--chemical synthesisPancreatic Elastase--antagonists & inhibitorsStructure-Activity RelationshipTime Factors