TY  - GEN
AU  - Asquith,Christopher R M
AU  - Tizzard,Graham J
AU  - Bennett,James M
AU  - Wells,Carrow I
AU  - Elkins,Jonathan M
AU  - Willson,Timothy M
AU  - Poso,Antti
AU  - Laitinen,Tuomo
TI  - Targeting the Water Network in Cyclin G-Associated Kinase (GAK) with 4-Anilino-quin(az)oline Inhibitors
SN  - 1860-7187
PY  - 2021///0614
KW  - Crystallography, X-Ray
KW  - Dose-Response Relationship, Drug
KW  - HEK293 Cells
KW  - Humans
KW  - Intracellular Signaling Peptides and Proteins
KW  - antagonists & inhibitors
KW  - Models, Molecular
KW  - Molecular Structure
KW  - Protein Kinase Inhibitors
KW  - chemical synthesis
KW  - Protein Serine-Threonine Kinases
KW  - Quinazolines
KW  - Structure-Activity Relationship
KW  - Water
KW  - chemistry
N1  - Publication Type: Journal Article; Research Support, Non-U.S. Gov't
UR  - https://doi.org/10.1002/cmdc.202000150
ER  -