The Lysosomotropic Activity of Hydrophobic Weak Base Drugs is Mediated via Their Intercalation into the Lysosomal Membrane. [electronic resource]
- Cells 04 2020
Publication Type: Journal Article
2073-4409
10.3390/cells9051082 doi
Antineoplastic Agents--pharmacology Cell Line, Tumor Central Nervous System Agents--analysis Drug Resistance, Neoplasm--drug effects Humans Hydrophobic and Hydrophilic Interactions--drug effects Intercalating Agents--analysis Intracellular Membranes Lysosomes--drug effects Molecular Dynamics Simulation Pharmaceutical Preparations--analysis Sequestering Agents--metabolism