Bahekar, Rajesh

Discovery of diaminopyrimidine-carboxamide derivatives as JAK3 inhibitors. [electronic resource] - Bioorganic chemistry 06 2020 - 103851 p. digital

Publication Type: Journal Article

1090-2120

10.1016/j.bioorg.2020.103851 doi


Animals
Antirheumatic Agents--chemical synthesis
Arthritis, Experimental--blood
Cell Line
Dose-Response Relationship, Drug
Drug Discovery
Humans
Janus Kinase 3--antagonists & inhibitors
Male
Mice
Mice, Inbred C57BL
Mice, Inbred DBA
Molecular Docking Simulation
Molecular Structure
Protein Kinase Inhibitors--chemical synthesis
Pyrimidines--chemical synthesis
Rats
Structure-Activity Relationship