Dong, Maoqing
Rational development of a high-affinity secretin receptor antagonist. [electronic resource]
- Biochemical pharmacology 07 2020
- 113929 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1873-2968
10.1016/j.bcp.2020.113929 doi
Alanine--metabolism
Amino Acid Sequence
Animals
Binding Sites
CHO Cells
Cricetulus
Drug Design
Glucagon-Like Peptide-1 Receptor--metabolism
Humans
Hydrophobic and Hydrophilic Interactions
Ligands
Models, Molecular
Peptides--chemistry
Protein Binding
Protein Conformation, alpha-Helical
Receptors, Calcitonin--metabolism
Receptors, G-Protein-Coupled--antagonists & inhibitors
Receptors, Gastrointestinal Hormone--antagonists & inhibitors
Secretin--analogs & derivatives