Dong, Maoqing

Rational development of a high-affinity secretin receptor antagonist. [electronic resource] - Biochemical pharmacology 07 2020 - 113929 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1873-2968

10.1016/j.bcp.2020.113929 doi


Alanine--metabolism
Amino Acid Sequence
Animals
Binding Sites
CHO Cells
Cricetulus
Drug Design
Glucagon-Like Peptide-1 Receptor--metabolism
Humans
Hydrophobic and Hydrophilic Interactions
Ligands
Models, Molecular
Peptides--chemistry
Protein Binding
Protein Conformation, alpha-Helical
Receptors, Calcitonin--metabolism
Receptors, G-Protein-Coupled--antagonists & inhibitors
Receptors, Gastrointestinal Hormone--antagonists & inhibitors
Secretin--analogs & derivatives