Beatty, Joel W

Discovery of Potent and Selective Non-Nucleotide Small Molecule Inhibitors of CD73. [electronic resource] - Journal of medicinal chemistry 04 2020 - 3935-3955 p. digital

Publication Type: Journal Article

1520-4804

10.1021/acs.jmedchem.9b01713 doi


5'-Nucleotidase--antagonists & inhibitors
Animals
Binding, Competitive--drug effects
CHO Cells
Cells, Cultured
Cricetinae
Cricetulus
Crystallography, X-Ray--methods
Drug Discovery--methods
GPI-Linked Proteins--antagonists & inhibitors
Hepatocytes--drug effects
Humans
Triazoles--chemistry