TY - GEN AU - Salomon,Emmanuel AU - Schmitt,Marjorie AU - Mouray,Elisabeth AU - McEwen,Alastair G AU - Bounaadja,Lotfi AU - Torchy,Morgan AU - Poussin-Courmontagne,Pierre AU - Alavi,Sarah AU - Tarnus,Céline AU - Cavarelli,Jean AU - Florent,Isabelle AU - Albrecht,Sébastien TI - Aminobenzosuberone derivatives as PfA-M1 inhibitors: Molecular recognition and antiplasmodial evaluation SN - 1090-2120 PY - 2021///0224 KW - Aminopeptidases KW - antagonists & inhibitors KW - Anisoles KW - chemical synthesis KW - Antimalarials KW - Cycloheptanes KW - Dose-Response Relationship, Drug KW - Enzyme Inhibitors KW - Molecular Structure KW - Parasitic Sensitivity Tests KW - Plasmodium falciparum KW - drug effects KW - Structure-Activity Relationship N1 - Publication Type: Journal Article; Research Support, Non-U.S. Gov't UR - https://doi.org/10.1016/j.bioorg.2020.103750 ER -