Qiu, Yunguang

TREK Channel Family Activator with a Well-Defined Structure-Activation Relationship for Pain and Neurogenic Inflammation. [electronic resource] - Journal of medicinal chemistry 04 2020 - 3665-3677 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1520-4804

10.1021/acs.jmedchem.9b02163 doi


Analgesics--metabolism
Animals
Anti-Inflammatory Agents--metabolism
Benzothiazoles--metabolism
Binding Sites
Ganglia, Spinal--drug effects
HEK293 Cells
Humans
Male
Mice, Inbred BALB C
Mice, Inbred C57BL
Molecular Docking Simulation
Molecular Structure
Neurogenic Inflammation--drug therapy
Pain--drug therapy
Pancreatitis--drug therapy
Potassium Channels, Tandem Pore Domain--agonists
Protein Binding
Rats, Sprague-Dawley
Structure-Activity Relationship