Mohareb, Rafat M

Heterocyclization of 2-(2-phenylhydrazono)cyclohexane-1,3-dione to Synthesis Thiophene, Pyrazole and 1,2,4-triazine Derivatives with Anti-Tumor and Tyrosine Kinase Inhibitions. [electronic resource] - Anti-cancer agents in medicinal chemistry 2020 - 1209-1220 p. digital

Publication Type: Journal Article

1875-5992

10.2174/1871520620666200310093911 doi


Antineoplastic Agents--chemical synthesis
Cell Line, Tumor
Cell Proliferation--drug effects
Cyclization
Dose-Response Relationship, Drug
Drug Screening Assays, Antitumor
Humans
Molecular Structure
Protein Kinase Inhibitors--chemical synthesis
Protein-Tyrosine Kinases--antagonists & inhibitors
Proto-Oncogene Proteins c-pim-1--antagonists & inhibitors
Pyrazoles--chemical synthesis
Structure-Activity Relationship
Thiophenes--chemical synthesis
Triazines--chemical synthesis