Targeting the Regulatory Site of ER Aminopeptidase 1 Leads to the Discovery of a Natural Product Modulator of Antigen Presentation. [electronic resource]
- Journal of medicinal chemistry 03 2020
- 3348-3358 p. digital
Publication Type: Journal Article
1520-4804
10.1021/acs.jmedchem.9b02123 doi
Allosteric Site Aminopeptidases--antagonists & inhibitors Animals Antigen Presentation--drug effects Catalytic Domain Crystallography, X-Ray Diterpenes, Clerodane--chemistry Enzyme Activators--chemistry Epitopes--chemistry HeLa Cells Humans Mice Minor Histocompatibility Antigens--chemistry Peptides--chemistry Protease Inhibitors--chemistry Protein Binding Proteolysis--drug effects