Liddle, John

Targeting the Regulatory Site of ER Aminopeptidase 1 Leads to the Discovery of a Natural Product Modulator of Antigen Presentation. [electronic resource] - Journal of medicinal chemistry 03 2020 - 3348-3358 p. digital

Publication Type: Journal Article

1520-4804

10.1021/acs.jmedchem.9b02123 doi


Allosteric Site
Aminopeptidases--antagonists & inhibitors
Animals
Antigen Presentation--drug effects
Catalytic Domain
Crystallography, X-Ray
Diterpenes, Clerodane--chemistry
Enzyme Activators--chemistry
Epitopes--chemistry
HeLa Cells
Humans
Mice
Minor Histocompatibility Antigens--chemistry
Peptides--chemistry
Protease Inhibitors--chemistry
Protein Binding
Proteolysis--drug effects