Le, Philipp

Repurposing human kinase inhibitors to create an antibiotic active against drug-resistant Staphylococcus aureus, persisters and biofilms. [electronic resource] - Nature chemistry 02 2020 - 145-158 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't; Research Support, U.S. Gov't, Non-P.H.S.

1755-4349

10.1038/s41557-019-0378-7 doi


Animals
Anti-Bacterial Agents--chemical synthesis
Autolysis--chemically induced
Benzodioxoles--chemical synthesis
Biofilms--drug effects
Cell Line, Tumor
Drug Repositioning
Female
Humans
Male
Methicillin-Resistant Staphylococcus aureus--drug effects
Mice, Inbred C57BL
Microbial Sensitivity Tests
Molecular Dynamics Simulation
Molecular Structure
Protein Kinase Inhibitors--chemistry
Sorafenib--analogs & derivatives
Structure-Activity Relationship