Singleton, Justin D

Synthesis and biological evaluation of novel pyrazolo[1,5-a]pyrimidines: Discovery of a selective inhibitor of JAK1 JH2 pseudokinase and VPS34. [electronic resource] - Bioorganic & medicinal chemistry letters 01 2020 - 126813 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1464-3405

10.1016/j.bmcl.2019.126813 doi


Class III Phosphatidylinositol 3-Kinases--antagonists & inhibitors
Humans
Janus Kinase 1--antagonists & inhibitors
Molecular Structure
Pyrimidines--chemical synthesis
Structure-Activity Relationship