Synthesis and biological evaluation of novel pyrazolo[1,5-a]pyrimidines: Discovery of a selective inhibitor of JAK1 JH2 pseudokinase and VPS34. [electronic resource]
- Bioorganic & medicinal chemistry letters 01 2020
- 126813 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1464-3405
10.1016/j.bmcl.2019.126813 doi
Class III Phosphatidylinositol 3-Kinases--antagonists & inhibitors Humans Janus Kinase 1--antagonists & inhibitors Molecular Structure Pyrimidines--chemical synthesis Structure-Activity Relationship